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DPA-713 or ''N'',''N''-diethyl-2-(4-methoxyphenyl)-5,7-dimethylpyrazolo()pyrimidine-3-acetamide is a selective ligand for the translocator protein (TSPO). The binding affinity of DPA-713 for TSPO is reported as ''K''i = 4.7 ± 0.2 nM. DPA-713 has been radiolabelled with carbon-11 as a potential radiotracer for imaging the TSPO using positron emission tomography (PET). Radiation dosimetry and biodistribution of ()DPA-713 have been assessed in healthy volunteers, indicating that ()DPA-713 is a suitable radioatracer for imaging the TSPO in humans. ==See also== * DPA-714 * translocator protein 抄文引用元・出典: フリー百科事典『 ウィキペディア（Wikipedia）』 ■ウィキペディアで「DPA-713」の詳細全文を読む スポンサード リンク
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